CP-409092-hydrochloride-DataSheet-生命科学试剂-MedChemExpress

1、Hotline: 400-820-3792Inhibitors Agonists Screening Librarieswww.MedChemECP-409092 hydrochlorideCat. No.: HY-101639ACAS No.: 225240-86-8分式: CHClNO分量: 333.81作靶点: GABA Receptor作通路: Membrane Transporter/Ion Channel; Neuronal Signaling储存式: Powder -20C 3 years4C 2 yearsIn solvent -80C 6 months-20C 1 month

2、溶解性数据体外实验 DMSO : 41.67 mg/mL (124.83 mM; Need ultrasonic)Mass Solvent1 mg 5 mg 10 mg Concentration制备储备液1 mM 2.9957 mL 14.9786 mL 29.9572 mL5 mM 0.5991 mL 2.9957 mL 5.9914 mL10 mM 0.2996 mL 1.4979 mL 2.9957 mL请根据产品在不同溶剂中的溶解度，选择合适的溶剂配制储备液，并请注意储备液的保存式和期限。体内实验 请根据您的实验动物和给药式选择适当的溶解案，配制前请先配制澄的储备液，再依次添加助溶剂

3、(为保证实验结果的可靠性，体内实验的作液，建议您现现配，当天使；澄的储备液可以根据储存条件，适当保存；以下溶剂前的百分指该溶剂在您配制终溶液中的体积占)：1. 请依序添加每种溶剂： 10% DMSO 40% PEG300 5% Tween-80 45% salineSolubility: 2.08 mg/mL (6.23 mM); Clear solution2. 请依序添加每种溶剂： 10% DMSO 90% (20% SBE-CD in saline)Solubility: 2.08 mg/mL (6.23 mM); Clear solution3. 请依序添加每种溶剂： 10% DMSO

4、 90% corn oilSolubility: 2.08 mg/mL (6.23 mM); Clear solution1/2 Master of Small Molecules 您边的抑制剂师www.MedChemEBIOLOGICAL ACTIVITY物活性 CP-409092 hydrochlorideGABAA 受体的部分激动剂，具有抗焦虑活性 1。REFERENCES1. Kamel A, et al. Metabolism, pharmacokinetics and excretion of the GABA(A) receptor partial agonist (14)CCP-409,092 in rats.Xenobiotica. 2010 Jun;40(6):400-14.McePdfHeightCaution: Product has not been fully validated for medical applications.For research use only.Tel: 400-820-3792;Fa