GPCR化合物库- Medchemexpress (MCE)

1、标题：GPCR化合物库- Medchemexpress （MCE）品牌： Medchemexpress （MCE）保存条件： -20供应商： MCE中国数量： 大量保质期： 2年规格：提供组合定制服务（现货供应）供货地址：美国     MedChemExpress (MCE)专注于各种抑制剂、调节剂、API、天然产物及化合物库，总部位于美国新泽西。MCE经过十年努力已成为全球生物活性小分子领域的一流供应商。MedChemExpress(MCE)产品涵盖近20个热门研究领域，1000多个细分靶点，超过3000个现货抑制剂、拮抗剂和激动剂。相关的应用成果已发表于Nat

2、ure、Cell等国际知名杂志，在全球20余个国家地区设有代理机构。上海皓元生物医药科技有限公司(MCE 中国) 是MedChemExpress (MCE) 亚洲总代理。  货号：HY-L006 A unique collection of 190 small molecules targeting G protein coupled receptors used in GPCR screening for various research and drug development projects. All of the small molecules in the GPCR li

3、brary are well characterized with biological and pharmaceutical activity. A powerful tool for discovering GPCR-based drugs that are the richest signal receptor targets for drug discovery. Targets such as 5-HT Receptor, Dopamine Receptor, Opioid Receptor, Adrenergic Receptors, Cannabinoid Receptor, m

4、GluR, and ETA-receptor etc. Structurally diverse, medicinally active, and cell permeable. Rich documentation with structure, IC50, and brief introduction. NMR and HPLC validated to ensure the highest purity.Formulation: A collection of 190 active molecules supplied as pre-dissolved DMSO solutio

5、nsContainer: 96 Well Format Sample Storage Tube With Screw Cap and Optional 2D BarcodeStability: 3 months -20°C in DMSO, 6 months -80°C in DMSOShipping: Blue icePackaging: Inert gasPlate layout: HY-EmptyAlosetron (Hydrochloride)AripiprazoleBRL 54443Clozapin

6、e N-oxideCP-809101 (hydrochloride)bEmptyOndansetron (hydrochloride dihydrate)Palonosetron (Hydrochloride)QuetiapineSB 271046 (Hydrochloride)SB-269970 (hydrochloride)cEmptyWAY-100635 (maleate salt)AdoprazineCapadenosonIstradefyllineLUF6000dEmptyHOKU-81ICI 118,551 (hydrochloride)IndacaterolIsoprenalin

7、e (hydrochloride)Ivabradine (hydrochloride)eEmptyTapentadol (hydrochloride)Angiotensin II humanAVE 0991AzilsartanAzilsartan medoxomil (monopotassium)fEmptyAM630JWH 073OtenabantRimonabant (Hydrochloride)TaranabantgEmptyINCB3344MK-0812MK-0974MK-3207 (Hydrochloride)OlcegepanthEmptySCH 527123SCH 546738S

8、CH 563705SRT3190WZ811789101112aLorcaserin (Hydrochloride)LoxapineLu AE58054 (Hydrochloride)LY 344864OlanzapineEmptybSB-742457SetiptilineTianeptineTropisetronVortioxetineEmptycPreladenantTozadenantAdipoRonCarvedilolFormoterol (Fumarate)EmptydMirabegronSalmeterol xinafoateSilodosinVilanterolAsenapineE

9、mptyeEprosartan (mesylate)OlmesartanOlmesartan medoxomilPD 123319 (ditrifluoroacetate)TelmisartanEmptyfWIN 55,212-2 (Mesylate)Calcium-Sensing Receptor Antagonists ICinacalcetNPS-2143NPS-2143 (hydrochloride)EmptygAMD-070 (hydrochloride)AMG 487NBI-74330PlerixaforReparixinEmptyhAMD 3465 (hexahydrobromi

10、de)Lurasidone (Hydrochloride)AmisulprideArmodafinilBrexpiprazoleEmptyPlate layout: HY-EmptyCariprazineHaloperidolPaliperidonerac-Rotigotine (Hydrochloride)RotigotinebEmptyBosentanMacitentanSitaxsentan (sodium)ZibotentanAnamorelincEmptyMK 0893BudesonideCortisone (acetate)DexamethasoneGlu

11、cocorticoid receptor agonistdEmptyGPR120 modulator 2GPR40 Activator 1GW-1100GW9508TAK-875eEmptyEbrotidineLoratadineMetiamidePitolisant (hydrochloride)ZaltidinefEmptyKi16425(R)-(+)-Tolterodine(R)-5-Hydroxymethyl TolterodineAclidinium (Bromide)CevimelinegEmptyUmeclidinium (bromide)VU0152100Xanomeline

12、(oxalate)CTEPDipragluranthEmptyVU 0357121GSK962040AprepitantNKP608SB-222200789101112aST-836 (hydrochloride)Ziprasidone (hydrochloride monohydrate)AmbrisentanAtrasentan (hydrochloride)AvosentanEmptybIbutamoren (Mesylate)Exendin-4glucagon receptor antagonists-1glucagon receptor antagonists-2glucagon r

13、eceptor antagonists-3EmptycTGR5 Receptor AgonistMK-6892GSK1292263MBX-2982GPR120 modulator 1EmptydTUG-770Bavisant (dihydrochloride hydrate)Bepotastine (Beslilate)Ciproxifan (maleate)Clemizole (hydrochloride)EmptyeFenspiride (Hydrochloride)Montelukast (sodium)AM095AM966Fingolimod (hydrochloride)Emptyf

14、DarifenacinDiphenmanil (methylsulfate)Solifenacin (hydrochloride)Tarafenacin (D-tartrate)Tiotropium (Bromide)EmptygLY341495LY404039mGlu2 agonistMPEP (Hydrochloride)MTEP (hydrochloride)EmptyhTalnetantML314ADL-5859Alvimopan (dihydrate)BAN ORL 24EmptyPlate layout: HY-EmptyCebranopadolJDTic

15、 (dihydrochloride)Meptazinol (hydrochloride)Methylnaltrexone (Bromide)Naloxone (hydrochloride)bEmptySuvorexantTCS 1102MRS 2578PrasugrelTicagrelorcEmptyProstaglandin E1SalirasibCCG-63802CCG-63808Siramesine (hydrochloride)dEmptyEmptyEmptyEmptyEmptyEmptyeEmptyEmptyEmptyEmptyEmptyEmptyfEmptyEmptyEmptyEmptyEmptyEmptygEmptyEmptyEmptyEmptyEmptyEmptyhEmptyEmptyEmptyEmptyEmptyEmpty789101112aNaltrexoneAlmorexant (hydrochloride)SB-334867 (free base)SB-408124SB-674042EmptybAH 6809LaropiprantMK-2894OC000459ONO-AE3-208Empty