Setiptiline-Org-8282-DataSheet-生命科学试剂-MedChemExpress

1、Hotline: 400-820-3792Inhibitors Agonists Screening Librarieswww.MedChemESetiptilineCat. No.: HY-32329CAS No.: 57262-94-9Synonyms: Org-8282分式: CHN分量: 261.36作靶点: 5-HT Receptor作通路: GPCR/G Protein; Neuronal Signaling储存式: Powder -20C 3 years4C 2 yearsIn solvent -80C 6 months-20C 1 month溶解性数据体外实验 DMSO : 2

2、5 mg/mL (95.65 mM; Need ultrasonic)H2O : 90% corn oilSolubility: 2.5 mg/mL (9.57 mM); Clear solution1/2 Master of Small Molecules 您边的抑制剂师www.MedChemEBIOLOGICAL ACTIVITY物活性 Setiptiline(Org-8282)为5羟胺受体拮抗剂。REFERENCES1. Yamada K, Furukawa T. Behavioral effects of a new antidepressant, setiptiline. Nihon

3、 Yakurigaku Zasshi. 1991 Jan;97(1):31-9.2. Kamimura M, Aoba A, Yamaguchi N et al. The effect of age on plasma level of setiptiline maleate in depressed patients. ProgNeuropsychopharmacol Biol Psychiatry. 1994 Oct;18(6):1015-26.3. Kuniyoshi M, Nakamura J, Miura C, Inanaga K. Effectiveness of concomit

4、ant setiptiline maleate (Tecipul) on negative symptoms ofschizophrenia. Prog Neuropsychopharmacol Biol Psychiatry. 1994 Mar;18(2):339-46.4. Niho T, Ito C, Shibutani Y, Hashizume H, Yamaguchi K. Pharmacological properties of MO-8282, a novel antidepressant. NihonYakurigaku Zasshi. 1986 Oct;88(4):309-20.McePdfHeightCaution: Product has not been fully validated for medical applications.For research use only.Tel: 400-820-3792;Fax: