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1、13章8章solutions溶液剂pharmaceutical excipients药物辅料solubility溶解度disintegration崩解diluted alcohol稀释乙醇dissolution溶出topical alcohol外用乙醇sublingual舌下的glycerin甘油buccal口腔黏膜的crude drugs原药vagmal阴道的ion-exchange离子交换punches冲dehydrate脱水dies模vehicle溶媒compressed tablets压制片solvents溶剂adjuncts辅料cosolvents潜溶剂diluents稀释剂hydr
2、oalcoholic醇水性质fillers填充剂ethanol酒精binders粘合剂organic compounds有机化合物adhesives粘合剂extraction提取disintegrants崩解剂reserve osmosis反渗透antiadherents抗粘剂menstruum溶媒glidants助流剂excipient赋形剂lubricants润滑剂insoluble不溶的colorants着色剂often preferred首选flavorants矫味剂flavorants矫味剂core核antimicrobial抗菌的shell壳preservatives防腐剂mult
3、iply compressed tablets多层片glycols丙二醇incompatibility禁忌parabens尼泊金类staged drug release阶段性释药the U.S. Food and Drug Administration(FDA)美国食品药品管理局sugarcoated tablets糖衣片over-the-counter(OTC)非处方药water soluble水溶性的diluted稀释的film-coated tablets薄膜片National Farmula(NF)国家处方集gastrointestinal胃肠的rubbing外用的enteric-co
4、ated tablets肠溶衣片color additives色素添加剂gastric mucosa胃肠粘膜perfume oils芳香油local effect局部作用bitter substances一点物质systemic absorption全身作用denarurant变性剂chewable tablets咀嚼片acetone丙酮effervescent tablets泡腾片abusive滥用的molded tablets模制片ingestion摄取,吸收triturates研碎物volatile挥发物,挥发的sucrose蔗糖flammable易燃的lactose乳糖tight co
5、ntainer气密容器pharmacist药师rubefacient发红剂immediate-release tablets速释片externally外部的,外表的modefied-release tablets控释片germicide杀菌剂extended/delaied/sustained-release tablets缓释片instruments仪器lyophilization冻干synonym等同于soft direct compression软直接压片法topical局部的the first-pass effect首过效应syrups糖浆剂quality standards质量标准c
6、oncentrated集中的,浓缩的compendial requirements一般要求nonmedicated非治疗用的engraved刻痕commercially available市售的weight vatiation片重差异pharmacist药师content uniformity含量均匀度pharmacy药学,药房thickness厚度therapeutic治疗的hardness硬度administering管理,实施disintegration崩解compatibility兼容性label claim标示量percolation过滤,浸透friability脆碎度elixirs
7、酏剂granulation颗粒palatability适口性,风味friabilator脆碎测定仪viscous黏的abrasion磨损adjunctive附加的,辅助的handle制备monographs专著package包装tinctures酊剂shipment运输thimerosal硫柳汞discharge释放microbial微生物的,细菌引起的body fluids体液precipitate沉淀,沉淀物,析出optimization最优化benzoin tincture安息香酊correlation相关性stopper塞子,胶塞quality assurance质量保证excessi
8、ve temperatures高温bioequivalence生物等效性photochemical光化学的new drug applications(NDAs)新药申报资料light-resist-ant containers避光容器permeability透过性camphorated tincture of opium樟脑的阿片酊剂wet granulation湿法制粒sprays喷雾剂dry granulation干法制粒spirits醑剂direct compression直接压片methods of extraction提取方法compressibility可压性maceration浸
9、渍damp mass制软材characterization性质screen过筛anti-cataract抗白内障microcrystalline cellulose微晶纤维素cyclodextrin环糊精croscarmellose交联羧甲纤维素eye drops眼药水alginic acid海藻酸contents目录povidone聚维酮transcorneal penetration跨角膜渗透cornstarch淀粉浆inclusion包合物glucose solution糖浆saline生理盐水methyl-cellulose甲基纤维素filter滤膜carboxymethylcellu
10、lose羟甲基纤维素power X-ray diffraction patterns粉末X射线衍射crumble破碎corneal角膜的thermostatical恒温的apparatus装置,设备humidity湿度permeability渗透性magnesium stearate硬脂酸镁calculation计算all-in-one granulation methods一步制粒法withdrawn取出the fluid bed granulator流化床制粒external water bath水浴acacia阿拉伯胶pharmacodynamics药效学hydroxypropyl ce
11、llulose羟丙基纤维素concentration浓度,集中moisture content湿度hereditary遗传的lower punch下冲biodegradable生物可降解的upper punch上冲matrices材料direct compression tableting粉末直接压片 microsphere微球spray-dried喷雾干燥properties性能,属性dioxide二氧化硅drug delivery system药物传递系统capping顶裂fabrication制造splitting裂片Wide-angle X-ray diffraction analys
12、is广角X射线衍射分析laminating分层phosphate buffered磷酸盐缓冲液entrapment包裹、陷入hardening rate硬化率fine power细粉drug ratio药物比,投料比physical deformations物理缺陷encapsulation efficiency包封率tablet dedusting片剂除尘crystallinity结晶度burst release突释conreolled release控释citrate枸橼酸14章15章immiscible不能混合dosage forms剂型dispersed phase分散相sterili
13、ty无菌dispersing phase分散介质microorganisms微生物dispersion medium分散介质irrigation冲洗dispersed system分散体系fluids流体miscible易混合的,能混溶的dialysis透析emulsification乳化作用vaccines疫苗fine droplets小液滴ophthalmic眼用的acrosol气溶胶pyrogen热原colloidal胶体的hypodermic皮下注射的dimension大小,尺寸buffers缓冲液coarse dispersions粗分散体added substances添加剂fin
14、e dispersions细分散体sterilization灭菌magmas胶浆剂steam蒸汽灭菌gels凝胶剂filtration滤过灭菌settle to the bottom沉降至瓶底performance性能uniform均一的,统一的autoclave高压灭菌moderate agitation温和搅拌microbial微生物ophthalmic眼用的denaturation变性otic耳用的adequate充分的sterile无菌的Percolation渗漉suspensions混悬剂sealed密闭的minimum最低的container容器solubility溶解度Ampul
15、(e)安瓿stabilizers稳定剂oleaginous油性的additives添加剂fixed oils不挥发油dilute稀释glycerin甘油aqueous水性的petrolatum凡士林reconstitution再分散paraffin石蜡therapy治疗commercially available市售的flexibility administration给药灵活度filter滤膜palatable气味宜人的pore size孔径chloramphenicol氯霉素specification规格taste-masking掩味millipore filter微孔滤膜pharmaci
16、st药师porosity孔隙率flavorants矫味剂retention截留affinity亲和性vacuum真空度penetrate渗透polar极性的clump together聚集literature文献hygroscopic吸湿性的filter assembly滤膜装置wetting agents润湿剂pyrogen testing热原检测displace取代、趋除、置换contamination污染penetration渗透endotoxins内毒素colloid mill胶体磨water for injection注射用水mortar乳钵nonvolatile不挥发的pestle
17、乳棒fractional distillation分馏soluble可溶的sytinges注射器colorant着色剂needles针头preservatives防腐剂interval间隔mixing equipment混合机械coagulate凝固uniformity均匀度threshold阈值bacterial细菌mold霉菌其他contamination污染hard gelatin capsules硬胶囊suspensoid混悬物hygroscopic吸湿的antacid抗酸剂desiccant干燥剂viscosity粘度activated charcoal活性炭homogenizer均
18、质机olintments软膏剂homomixer均匀混合器,高速搅拌机creams乳膏剂sustained-release缓释gels凝胶剂compound fomulation复方carboxymethycellulose羧甲基纤维素stability稳定性hydroxypropyl methylcellulose羟丙甲纤维素matrix基质tragacanth西黄蓍胶microencapsulation微囊化pastes涂剂ion exchange resins离子交换树脂plasters橡皮膏complex复合物Vanishing cream雪花膏gastrointestinal tra
19、ct胃肠道edetate disodiumEDTAemulsifying agents乳化剂suppositories栓剂emulsifier乳化剂inserts塞入剂be compatible with与配伍、相容formulative ingredients成分组分上接14章interfere干扰olive oil橄榄油therapeutic agent治疗剂calamine炉甘石deteriorate变质、腐败biphasic二相capability能力、性能transdermal透明的 经皮的carbohydrate碳水化合物artificial人工的acacia阿拉伯胶aggrega
20、tion and coalescence聚集和合并tragacanth西黄蓍胶creaming乳液分层agar琼脂reversible process可逆过程pectin果胶alternative test交错实验thickening agents增稠剂antioxidants抗氧化剂microcrystalline微晶纤维素sol溶胶viscosity regulator粘度调节剂aerosol气溶胶settling沉降opaques不透明的gelatin明胶unigorm不均匀的eggyolk蛋黄lyophilic亲液的lotions洗剂lyophobic疏液的ointments软膏剂hy
21、drophilic亲水的cholesterol胆固醇hydrophobic疏水的derivatives衍生物association结合、联合anionic阴离子amphiphilic colloid两性的cationic阳离子semisolid半固体nonionic非离子thixotropy触变性grinding研磨micropulverizer微粉化(机)triturate研磨oleic acid油酸graduate量筒insuincient不够的swirl漩涡、打旋occlusion封闭as is deemed根据需要in situ soap method新生皂法auxiliary辅助的t
22、hickness厚度mannitol甘露醇sublingual舌下sucrose蔗糖Buccal口腔黏膜lactose乳糖Vaginal阴道lyophilization冻干compressed tablets压制片excipients赋形剂multiply compressed tablets多层压制片weight variation重量差异Sugarcoated tablets糖包衣片content uniformity含量均匀度Film-coated tablets薄膜包衣片thickness厚度Enteric-coated tablets肠溶衣片friability脆碎度Chewable
23、 tablets咀嚼片tablet dissolution溶出度Effervescent tablets泡腾片wet/dry granulation湿法/干法制粒Dispensing tablets分散片direct compression直接压片法Hypodermic tablets植入片excipients辅料Immediate-release tablets速释片magnesium stearate硬脂酸镁Buccal and sublingual tablets口腔和舌下片talc滑石粉Instantly disintegrating or dissolving tablets 快速崩
24、解或溶出片All-in-one granulation methods一步制粒法extended-release tablets缓释片fluid bed流化床Punches and dies冲和模acacia阿拉伯胶diluents (fillers)稀释剂lactose乳糖binders (adhesives)黏合剂maltose麦芽糖disintegrants崩解剂mannitol甘露醇antiadherents抗粘剂sorbitol山梨醇glidants助流剂dextrose右旋糖酐lubricants润滑剂xylitol木糖醇chemical or physical incompati
25、bility化学或物理不相容性humidity湿度delayed-release迟释片hygroscopic吸湿的disintegrate崩解desiccant干燥剂dissolution 溶出activated charcoal活性炭absorption吸收fasting禁食effect起效enteric coating肠溶包衣 Starch淀粉Solid dispersions固体 分散体shellac虫胶colloidal胶体的ointments软膏uniform均一的creams霜剂,乳剂ophthalmic眼科的thixotrope触变胶affinity亲和性methylparabe
26、n尼泊金甲酯Penetration, permeability渗透 , 渗透性propylparaben尼泊金丙酯mortar研钵vagina阴道colloid mill, fluid energy mill胶体磨流能磨rectum直肠viscosity粘度suppositories栓剂dispersion分散体系inserts塞入剂oleaginous油性的distillation method蒸馏法emulsifying agent乳化剂ion exchange method离子交换法lotions洗液reverse osmosis反渗透liniments擦剂sodium citrate枸
27、橼酸钠coalesce合并syrups糖浆剂Hydrophile-Lipophile Balance HLB亲水亲油平衡值solubility(汉译英)溶解度precipitating沉淀作用stability稳定性proportions比例bioavailibility生物利用度in situ soap method新生皂法compatibility相容性考:干胶、湿胶法制备viscous粘性的oleic acid油酸monographs专著microemulsions微乳tinctures醑剂aggregation and coalescence聚集与合并thimerosal硫柳汞micr
28、ocrystalline cellulose微晶纤维素glycerin甘油sol溶胶stopper塞子opaques遮光剂maceration浸渍lyophilic亲液的percolation渗漉lyophobic疏液的Emulsification乳化hydrophilic亲水的aerosol气雾剂、气溶胶hydrophobic疏水的amphiphilic两亲的intramuscular IM肌肉内micropulverizer微粉化intradermal ID皮内propellant抛射剂P.O口服inhalation吸入buffer缓冲液sprays喷雾preservatives防腐剂di
29、sinfectants消毒剂steam sterilization蒸汽灭菌sterility无菌autoclave灭菌锅ig灌胃gauges计量表irrigation冲洗剂community pharmacy社区药房dialysis透析ophthalmic preparations眼用制剂intravenous IV静脉内的练习重点 汉译英国家食品药品监督管理局SFDA多层片multilayer tablet纳米制剂nanometer preparatation胃液gastric juice16目-筛16 mesh screen高压蒸汽灭菌high pressure steam sterili
30、zation肠衣片enteric coated tablets剂型dosage forms渗漉percolate混悬剂suspensions药剂学pharmaceutics脂肪乳fat emulsion首过效应first pass effect量筒graduated flask粒密度particle density输液transfusion粒度分布size distribution溶出实验dissolution test乳剂emulsions小丸pellets微球microsphere热原检测pyrogen test软胶囊soft gelatin capsules制粒granulation中国药典Ch.P
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